Items where Author is "Docsa, Tibor"

Article

Homolya, Levente, Mathomes, Rachel Thelma ORCID: 0000-0002-1079-8509, Varga, Luca, Docsa, Tibor, Juhasz, Laszlo, Hayes, Joseph ORCID: 0000-0002-7745-9616 and Somsák, László (2024) Synthesis, in silico and kinetics evaluation of N-(β-D-glucopyranosyl)-2-arylimidazole-4(5)-carboxamides and N-(β-D-glucopyranosyl)-4(5)-arylimidazole-2-carboxamides as glycogen phosphorylase inhibitors. International Journal of Molecular Sciences, 25 (9). ISSN 1661-6596

Kun, Sándor, Mathomes, Rachel Thelma ORCID: 0000-0002-1079-8509, Docsa, Tibor, Somsák, László and Hayes, Joseph ORCID: 0000-0002-7745-9616 (2023) Design and Synthesis of 3-(β-d-Glucopyranosyl)-4-amino/4-guanidino Pyrazole Derivatives and Analysis of Their Glycogen Phosphorylase Inhibitory Potential. Molecules, 28 (7). p. 3005.

Barr, Daniel, Szennyes, Eszter, Bokor, Éva, Al-Oanzi, Ziad H., Moffatt, Colin, Kun, Sándor, Docsa, Tibor, Sipos, Ádám, Davies, Matthew et al (2019) Identification of C-β-d-Glucopyranosyl Azole-Type Inhibitors of Glycogen Phosphorylase That Reduce Glycogenolysis in Hepatocytes: In Silico Design, Synthesis, in Vitro Kinetics, and ex Vivo Studies. ACS Chemical Biology, 14 (7). pp. 1460-1470. ISSN 1554-8929

Kun, Sándor, Begum, Jaida, Kyriakis, Efthimios, Stamati, Evgenia C V, Barkas, Thomas A, Szennyes, Eszter, Bokor, Éva, Szabó, Katalin E, Stravodimos, George A et al (2018) A multidisciplinary study of 3-(β-d-glucopyranosyl)-5-substituted-1,2,4-triazole derivatives as glycogen phosphorylase inhibitors: Computation, synthesis, crystallography and kinetics reveal new potent inhibitors. European Journal of Medicinal Chemistry, 147 . pp. 266-278. ISSN 0223-5234

Begum, Jaida, Varga, Gergely, Docsa, Tibor, Gergely, Pál, Hayes, Joseph M. ORCID: 0000-0002-7745-9616, Juhász, László and Somsák, László (2015) Computationally motivated synthesis and enzyme kinetic evaluation of N-(β-d-glucopyranosyl)-1,2,4-triazolecarboxamides as glycogen phosphorylase inhibitors. Med. Chem. Commun., 6 (1). pp. 80-89. ISSN 2040-2503